GR 231118

GR 231118 is a potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively), and also a NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively).

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CAT#R0829
CAS158859-98-4
M.F/FormulaC110H170N34O24
M.W/Mr.2352.77
SequenceIEPXYRLRY IEPXYRLRY*(Modifications: X = Dpr, Amide Bridge = 2 - 4*, 4 - 2*, Tyr-9 = C-terminal amide)
Labeling TargetNeuropeptide Y (NPY) Y1 receptor
ApplicationA potent NPY1-R antagonist and NPY4-R agonist
AppearanceWhite lyophilised solid
Purity>99 %
ActivityAntagonist
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