K-(D-1-Nal)-FwLL-NH2 is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively), which blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
CAT# | R0816 |
CAS | 1394288-22-2 |
M.F/Formula | C51H67N9O6 |
M.W/Mr. | 902.13 |
Sequence | KXFWLL(Modifications: X=D-1-Nal,Trp-4 = D-Trp, Leu-6 = C-terminal amide) |
Labeling Target | Ghrelin receptor |
Application | K-(D-1-Nal)-FwLL-NH2 is an inverse agonist of the ghrelin receptor. |
Purity | >98 % |
Activity | Agonist |
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