A highly selective, potent antagonist for the opioid δ-receptor. It exhibits partial agonist in vitro activity at δ receptors at high concentrations.
CAT# | R1076 |
CAS | 89352-67-0 |
Synonyms/Alias | N,N-Di-2-propen-1-yl-L-tyrosyl-2-methylalanyl-L-phenylalanyl-L-leucine; NIH 10893 |
M.F/Formula | C38H53N5O7 |
M.W/Mr. | 691.87 |
Sequence | YXXFL(Modifications: Tyr-1 = N,N-diallyl-Tyr, X = Aib) |
Labeling Target | Opioid Receptor |
Appearance | White lyophilised solid |
Purity | >98% |
Activity | Antagonist |
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