CYT-1010

CYT-1010 is an μ-opioid receptor ligand potentially for the treatment of acute and chronic pain and neuropathic pain syndrome.

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CAT#	10-101-237
Chemical Structure
CAS	213769-33-6
Synonyms/Alias	CYT1010, CYT 1010
Chemical Name	2-amino-N-[3-benzyl-6-(1H-indol-3-ylmethyl)-2,5,8-trioxo-1,4,7-triazacyclotridec-9-yl]-3-(4-hydroxyphenyl)propanamide
M.F/Formula	C35H40N6O5
M.W/Mr.	624.73
Application	Acute and chronic pain and neuropathic pain syndrome
Appearance	Solid powder
Activity	Agonist
Biological Activity	CYT-1010 is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively.

CAT#	Product Name	Inquiry
10-101-264	c(phg-isoDGR-(NMe)k)	Inquiry
10-101-127	Xipamide	Inquiry
10-101-284	[Ala1,3,11,15]-Endothelin 1	Inquiry
10-101-271	Biotin-Amylin (1-37), human amidated	Inquiry
HB00136	4-Oxothiane	Inquiry

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Storage	Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility	Soluble in DMSO
Shipping Condition	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
InChI	InChI=1S/C35H40N6O5/c36-27(18-23-13-15-25(42)16-14-23)32(43)39-29-12-6-7-17-37-33(44)30(19-22-8-2-1-3-9-22)40-35(46)31(41-34(29)45)20-24-21-38-28-11-5-4-10-26(24)28/h1-5,8-11,13-16,21,27,29-31,38,42H,6-7,12,17-20,36H2,(H,37,44)(H,39,43)(H,40,46)(H,41,45)
InChI Key	CFVGCGXJRNVTFP-UHFFFAOYSA-N
Canonical SMILES	C1CCNC(=O)C(NC(=O)C(NC(=O)C(C1)NC(=O)C(CC2=CC=C(C=C2)O)N)CC3=CNC4=CC=CC=C43)CC5=CC=CC=C5
References	1. Theodore E. Maione, Novel therapeutic uses of mu-opiate receptor peptides. WO2013173730A2.